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Eva Estébanez-Perpiñá
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A surface on the androgen receptor that allosterically regulates coactivator binding
E Estébanez-Perpiñá, LA Arnold, P Nguyen, ED Rodrigues, E Mar, ...
Proceedings of the National Academy of Sciences 104 (41), 16074-16079, 2007
3492007
The molecular mechanisms of coactivator utilization in ligand-dependent transactivation by the androgen receptor
E Estébanez-Perpiná, JMR Moore, E Mar, E Delgado-Rodrigues, ...
Journal of Biological Chemistry 280 (9), 8060-8068, 2005
2032005
Structure of the homodimeric androgen receptor ligand-binding domain
M Nadal, S Prekovic, N Gallastegui, C Helsen, M Abella, K Zielinska, ...
Nature communications 8 (1), 14388, 2017
1792017
Nuclear receptor crosstalk — defining the mechanisms for therapeutic innovation
K De Bosscher, SJ Desmet, D Clarisse, E Estébanez-Perpiña, ...
Nature Reviews Endocrinology, 2020
1542020
EPI-001, a compound active against castration-resistant prostate cancer, targets transactivation unit 5 of the androgen receptor.
SX De Mol E, Fenwick RB, Phang CT, Buzon V, Szulc E, De La Fuente A ...
ACS Chem Biol, 2016
133*2016
Discovery of small molecule inhibitors of the interaction of the thyroid hormone receptor with transcriptional coregulators
LA Arnold, E Estébanez-Perpiñá, M Togashi, N Jouravel, A Shelat, ...
Journal of Biological Chemistry 280 (52), 43048-43055, 2005
1322005
A conserved surface on the ligand binding domain of nuclear receptors for allosteric control
V Buzón, LR Carbó, SB Estruch, RJ Fletterick, E Estébanez-Perpiñá
Molecular and cellular endocrinology 348 (2), 394-402, 2012
922012
Crystal structure of the caspase activator human granzyme B, a proteinase highly specific for an Asp-P1 residue
E Estébanez-Perpiñá, P Fuentes-Prior, D Belorgey, M Braun, ...
Walter de Gruyter 381 (12), 1203-1214, 2000
842000
Structural insight into the mode of action of a direct inhibitor of coregulator binding to the thyroid hormone receptor
E Estebanez-Perpina, LA Arnold, N Jouravel, M Togashi, J Blethrow, ...
Molecular Endocrinology 21 (12), 2919-2928, 2007
762007
Advances in our structural understanding of orphan nuclear receptors
N Gallastegui, JAG Mackinnon, RJ Fletterick, E Estébanez-Perpiñá
Trends in biochemical sciences 40 (1), 25-35, 2015
732015
Allosteric conversation in the androgen receptor ligand-binding domain surfaces
S Grosdidier, LR Carbó, V Buzón, G Brooke, P Nguyen, JD Baxter, ...
Molecular Endocrinology 26 (7), 1078-1090, 2012
712012
The 2.2-Å crystal structure of human pro-granzyme K reveals a rigid zymogen with unusual features
C Hink-Schauer, E Estébanez-Perpiná, E Wilharm, P Fuentes-Prior, ...
Journal of Biological Chemistry 277 (52), 50923-50933, 2002
712002
Coregulator control of androgen receptor action by a novel nuclear receptor-binding motif
K Jehle, L Cato, A Neeb, C Muhle-Goll, N Jung, EW Smith, V Buzon, ...
Journal of Biological Chemistry 289 (13), 8839-8851, 2014
672014
Crystal structure of the apoptosis-inducing human granzyme A dimer
C Hink-Schauer, E Estébanez-Perpiñá, FC Kurschus, W Bode, DE Jenne
Nature Structural & Molecular Biology 10 (7), 535-540, 2003
672003
Effects of adult dysthyroidism on the morphology of hippocampal neurons
J Sala-Roca, E Estebanez-Perpina, F Balada, A Garau, ...
Behavioural brain research 188 (2), 348-354, 2008
542008
Inhibitors of the interaction of a thyroid hormone receptor and coactivators: preliminary structure− activity relationships
LA Arnold, A Kosinski, E Estébanez-Perpiñá, RK Guy
Journal of medicinal chemistry 50 (22), 5269-5280, 2007
542007
Regulation of androgen receptor activity by transient interactions of its transactivation domain with general transcription regulators
E De Mol, E Szulc, C Di Sanza, P Martínez-Cristóbal, CW Bertoncini, ...
Structure 26 (1), 145-152. e3, 2018
522018
Crystal structure of a novel mid-gut procarboxypeptidase from the cotton pest Helicoverpa armigera
E Estébanez-Perpiñá, A Bayés, J Vendrell, MA Jongsma, DP Bown, ...
Journal of molecular biology 313 (3), 629-638, 2001
482001
Oleic acid is an endogenous ligand of TLX/NR2E1 that triggers hippocampal neurogenesis
P Kandel, F Semerci, R Mishra, W Choi, A Bajic, D Baluya, LH Ma, ...
Proceedings of the National Academy of Sciences (PNAS) 119 (13), e2023784119, 2022
392022
Glucocorticoid Resistance: Interference between the Glucocorticoid Receptor and the MAPK Signalling Pathways
LM Sevilla, A Jiménez-Panizo, A Alegre-Martí, E Estébanez-Perpiñá, ...
International Journal of Molecular Sciences 22 (18), 10049, 2021
392021
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