Discovery of new cholesteryl ester transfer protein inhibitors via ligand-based pharmacophore modeling and QSAR analysis followed by synthetic exploration R Abu Khalaf, GA Sheikha, Y Bustanji, MO Taha European journal of medicinal chemistry 45 (4), 1598-1617, 2010 | 69 | 2010 |
Molecular modeling based approach, synthesis, and cytotoxic activity of novel benzoin derivatives targeting phosphoinostide 3-kinase (PI3Kα) DA Sabbah, M Saada, R Abu Khalaf, S Bardaweel, K Sweidan, T Al-Qirim, ... Bioorganic & medicinal chemistry letters 25 (16), 3120-3124, 2015 | 39 | 2015 |
Benzoin Schiff Bases: Design, Synthesis, and Biological Evaluation as Potential Antitumor Agents DA Sabbah, F Al-Tarawneh, WH Talib, K Sweidan, SK Bardaweel, ... Medicinal Chemistry 14 (7), 695 - 708, 2018 | 25 | 2018 |
Discovery of New Antifungal Leads via Pharmacophore Modeling and QSAR Analysis of Fungal N‐Myristoyl Transferase Inhibitors Followed by In Silico Screening MO Taha, AM Qandil, T Al‐Haraznah, R Abu Khalaf, H Zalloum, ... Chemical biology & drug design 78 (3), 391-407, 2011 | 25 | 2011 |
Design, synthesis, and biological evaluation of benzylamino-methanone based cholesteryl ester transfer protein inhibitors GA Sheikha, R Abu Khalaf, A Melhem, G Albadawi Molecules 15 (8), 5721-5733, 2010 | 25 | 2010 |
In Vivo Antihyperlipidemic Activity of a New Series of N‐(Benzoylphenyl) and N‐(Acetylphenyl)‐1‐benzofuran‐2‐carboxamides in Rats T Al‐Qirim, G Shattat, K Sweidan, W El‐Huneidi, GA Sheikha, ... Archiv der Pharmazie 345 (5), 401-406, 2012 | 23 | 2012 |
Exploring natural products as a source for antidiabetic lead compounds and possible lead optimization R Abu Khalaf Current Topics in Medicinal Chemistry 16 (23), 2549-2561, 2016 | 22 | 2016 |
Structure-Based Design: Synthesis, X-Ray Crystallography, and Biological Evaluation of N-Substituted-4-Hydroxy-2-Quinolone-3-Carboxamides as Potential PI3Kα Inhibitors D Sabbah, B Hishmah, K Sweidan, S Bardaweel, M AlDamen, H Zhong, ... Anti-Cancer Agents in Medicinal Chemistry 18 (2), 263-276, 2017 | 21 | 2017 |
Discovery of new β-D-glucosidase inhibitors via pharmacophore modeling and QSAR analysis followed by in silico screening R Abu Khalaf, AM Abdula, MS Mubarak, MO Taha Journal of molecular modeling 17 (3), 443-464, 2011 | 21 | 2011 |
Discovery of new β‐D‐galactosidase inhibitors via pharmacophore modeling and QSAR analysis followed by in silico screening AM Abdula, R Abu Khalaf, MS Mubarak, MO Taha Journal of computational chemistry 32 (3), 463-482, 2011 | 20 | 2011 |
Molecular docking and pharmacophore modeling studies of fluorinated benzamides as potential CETP inhibitors R Abu Khalaf, S Al-Rawashdeh, D Sabbah, G Abu Sheikha Medicinal Chemistry 13 (3), 239-253, 2017 | 18 | 2017 |
Design, synthesis, and biological evaluation of sulfonic acid ester and benzenesulfonamide derivatives as potential CETP inhibitors R Abu Khalaf, GA Sheikha, M Al-Sha’er, G Albadawi, M Taha Medicinal Chemistry Research 21 (11), 3669-3680, 2012 | 16 | 2012 |
Tryptophan and thiosemicarbazide derivatives: design, synthesis, and biological evaluation as potential β-d-galactosidase and β-d-glucosidase inhibitors R Abu Khalaf, AM Abdula, MS Mubarak, MO Taha Medicinal Chemistry Research 24 (6), 2529-2550, 2015 | 12 | 2015 |
Pharmacophore modeling and molecular docking studies of acridines as potential DPP-IV inhibitors R Abu Khalaf, Z Jarekji,T Al-Qirim, D Sabbah, G Shattat Canadian Journal of Chemistry 93 (7), 721-729, 2015 | 12 | 2015 |
Synthesis, biological evaluation and molecular modeling study of substituted benzyl benzamides as CETP inhibitors R Abu Khalaf, D Sabbah, E Al-Shalabi, S Bishtawi, G Albadawi, ... Archiv der Pharmazie 350 (12), 1-14, 2017 | 11 | 2017 |
CETP Inhibitory Activity of Chlorobenzyl Benzamides: QPLD Docking, Pharmacophore Mapping, and Synthesis R Abu Khalaf, H Abd El-Aziz, D Sabbah, G Albadawi, G Abu Sheikha Letters in Drug Design & Discovery 14 (12), 1391-1400, 2017 | 11 | 2017 |
Design, Synthesis and Biological Evaluation of N4-Sulfonamido-Succinamic, Phthalamic, Acrylic and Benzoyl Acetic Acid Derivatives as Potential DPP IV Inhibitors R Abu Khalaf, GA Sheikha, M Al-Sha'er, M Taha The open medicinal chemistry journal 7, 39-48, 2013 | 11 | 2013 |
Ligand-Based Drug Design: Synthesis and Biological Evaluation of Substituted Benzoin Derivatives as Potential Antitumor Agents. DA Sabbah, AH Ibrahim, WH Talib, KM Alqaisi, K Sweidan, SK Bardaweel, ... Medicinal chemistry (Shariqah (United Arab Emirates)) 15 (4), 417-429, 2019 | 10 | 2019 |
Isolation and Structure Elucidation of Bioactive Polyphenols R Abu Khalaf, A Alhusban, E Al-Shalabi, I Al-Sheikh, D Sabbah Studies in Natural Product Chemistry (Bioactive Natural Products) 63, 267-337, 2019 | 9* | 2019 |
Synthesis, Structural Characterization and Docking Studies of Sulfamoyl-Phenyl Acid Esters as Dipeptidyl Peptidase-IV Inhibitors R Abu Khalaf, D Sabbah, E Al-Shalabi, I Al-Sheikh, G Albadawi, ... Current Computer-Aided Drug Design 14 (2), 142-151, 2018 | 9 | 2018 |